Design and enantioselective synthesis of chiral pyranone fused indole derivatives with antibacterial activities against Xanthomonas oryzae pv oryzae for protection of rice

• Main Authors: Teng, Kunpeng, Liu, Qian, Zhang, Meng, Naz, Hira, Zheng, Pengcheng, Wu, Xingxing, Chi, Robin Yonggui
• 其他作者: School of Chemistry, Chemical Engineering and Biotechnology
• 格式: Article
• 語言: English
• 出版: 2024
• 主題: Agricultural Sciences; Chiral indole derivatives; Bacterial activity
• 在線閱讀: https://hdl.handle.net/10356/174249

A new class of chiral pyranone fused indole derivatives were prepared by means of N-heterocyclic carbene (NHC) organocatalysis and demonstrated notable antibacterial activity against Xanthomonas oryzae pv oryzae (Xoo). Bioassays showed that compounds (3S,4R)-5b, (3S,4R)-5d, and (3S,4R)-5l exhibited...