Mechanism-based inactivation of CYP450 enzymes: A case study of lapatinib

Mechanism-based inactivation of CYP450 enzymes: A case study of lapatinib

10.3109/03602532.2014.1003648

Saved in:

書目詳細資料
Main Authors:	Ho, Han Kiat, Chan, James Chun Yip, Hardy, Klarissa D., Chan, Eric Chun Yong
其他作者:	PHARMACY
格式:	Review
語言:	English
出版:	Informa Healthcare 2015
在線閱讀:	http://scholarbank.nus.edu.sg/handle/10635/120529
標簽:	添加標簽沒有標簽, 成為第一個標記此記錄!

相似書籍

Mechanism-based inactivation of CYP450 enzymes: A case study of lapatinib
由: Ho H.K, et al.
出版: (2016)

Mechanism-based inactivation of cytochrome P450 3A4 by lapatinib
由: Teng, W.C., et al.
出版: (2014)

Interaction of lapatinib with cytochrome P450 3A5
由: Chan, E.C.Y., et al.
出版: (2014)

Effect of CYP3A4 inducer dexamethasone on hepatotoxicity of lapatinib: Clinical and in vitro evidence
由: Teo, Y.L., et al.
出版: (2014)

Computational studies of the mechanisms of chemical reactions involved in mechanism-based inactivation of cytochrome P450 enzymes
由: Chuanprasit, Pratanphorn
出版: (2017)

Metabolic intermediate complex formation of human cytochrome P450 3A4 by lapatinib
由: Takakusa, H., et al.
出版: (2014)

Inhibitory effects of Thai herbal extracts on the cytochrome P450 3A-mediated the metabolism of gefitinib, lapatinib and sorafenib
由: Rodseeda C.
出版: (2023)

Upregulation of CYP 450s expression of immortalized hepatocyte-like cells derived from mesenchymal stem cells by enzyme inducers
由: Khanit Sa-ngiamsuntorn, et al.
出版: (2018)

Upregulation of CYP 450s expression of immortalized hepatocyte-like cells derived from mesenchymal stem cells by enzyme inducers
由: Khanit Sa-ngiamsuntorn, et al.
出版: (2017)

TRANSIENT TRANSFORMATION OF THE GENE ENCODING CYTOCHROME P450 MONOOXYGENASE ENZYME (CYP71AV1) INTO ARTEMISIA ANNNUA L.
由: Sulfiani Saula, Lely

Cloning and expression of Anopheles minimus NADPH-Cytochrome P450 reductase gene and in Vitro study of CYP6P7 enzyme system
由: Dolnapa Kaewpa
出版: (2023)

Mechanism-based inactivation of cytochrome P450 2A6 and 2A13 by Rhinacanthus nasutus constituents
由: Phisit Pouyfung, et al.
出版: (2018)

Effects of Cannabidiol and Δ9-tetrahydrocannabinol on Cytochrome P450 Enzymes: A Systematic Review
由: Sarah Smith, et al.
出版: (2024)

Cloning of cytochrome P450, CYP6P5, and CYP6AA2 from Anopheles minimus resistant to deltamethrin
由: Pornpimol Rongnoparut, et al.
出版: (2018)

Importance of H-abstraction in the final step of nitrosoalkane formation in the mechanism-based inactivation of cytochrome P450 by amine-containing drugs
由: Xu, Kai, et al.
出版: (2014)

Optimizing bacterial expression of catalytically active human cytochromes P450: Comparison of CYP2C8 and CYP2C9
由: S. L. Boye, et al.
出版: (2018)

Pivotal role of water in terminating enzymatic function : a density functional theory study of the mechanism-based inactivation of cytochromes P450
由: Hirao, Hajime, et al.
出版: (2013)

Reversible time-dependent inhibition of cytochrome P450 enzymes by duloxetine and inertness of its thiophene ring towards bioactivation
由: Chan, C.Y., et al.
出版: (2014)

Effects of curcuma comosa roxb. Extract on the expression of cyp450s in immortalized hepatocyte-like cells (imhc)
由: Petdao Petchuay, et al.
出版: (2022)

CYP5122A1, a novel cytochrome P450 is essential for survival of Leishmania donovani
由: Verma S., et al.
出版: (2019)

Lapatinib sensitivity in nasopharyngeal carcinoma is modulated by SIRT2-mediated FOXO3 deacetylation
由: Sathid Aimjongjun, et al.
出版: (2020)

Variable inhibitory effect of herbal supplements of different brands on human P450 CYP1A2
由: Sompon Wanwimolruk, et al.
出版: (2018)

Cytochrome P450 enzyme : its clinical role in drug interactions
由: Pailin Ujjin, et al.
出版: (2006)

EVOLVING ENANTIOSELECTIVE P450 MONOOXYGENASE FOR BIOHYDROXYLATIONS WITH MICROFLUIDIC ENZYME SCREENING
由: LIN YI
出版: (2024)

How Is a metabolic intermediate formed in the mechanism-based inactivation of cytochrome P450 by using 1,1-dimethylhydrazine : hydrogen abstraction or nitrogen oxidation?
由: Hirao, Hajime, et al.
出版: (2014)

METABOLIC ACTIVATION OF FIBROBLAST GROWTH FACTOR RECEPTOR INHIBITORS BY CYTOCHROME P450: MECHANISTIC INVESTIGATIONS INTO THE BIOCHEMICAL BASIS AND PHARMACOKINETIC IMPLICATIONS OF MECHANISM-BASED INACTIVATION
由: TANG WEI TAT LLOYD
出版: (2022)

Quantitative Proteomics-based Bottom-up PBK Modeling: A Case Study of 3 Statins
由: CHAN, JAMES CHUN YIP, et al.
出版: (2019)

Inhibitory effects of phyllanthus amarus and its major lignans on human microsomal cytochrome P450 activities: Evidence for CYP3A4 mechanism-based Inhibition
由: Theerada Taesotikul, et al.
出版: (2018)

Cytochrome P450 enzyme mediated herbal drug interactions (Part 2)
由: Sompon Wanwimolruk, et al.
出版: (2018)

Cytochrome P450 enzyme mediated herbal drug interactions (part 1)
由: Sompon Wanwimolruk, et al.
出版: (2018)

WRKY9 transcription factor regulates cytochrome P450 genes CYP94B3 and CYP86B1, leading to increased root suberin and salt tolerance in Arabidopsis
由: Krishnamurthy, Pannaga, et al.
出版: (2023)

Mechanism-based inhibition of cytochrome P450 3A4 by therapeutic drugs
由: Zhou, S., et al.
出版: (2014)

Functional polymorphisms of the cytochrome P450 1A2 (CYP1A2) gene and prolonged QTc interval in schizophrenia
由: Tay, J.K.X., et al.
出版: (2011)

Application of support vector machines to in silico prediction of cytochrome P450 enzyme substrates and inhibitors
由: Yap, C.W., et al.
出版: (2014)

Allele frequencies of single nucleotide polymorphisms of clinically important drug-metabolizing enzymes CYP2C9, CYP2C19, and CYP3A4 in a Thai population
由: Rattanaporn Sukprasong, et al.
出版: (2022)

Synergy between rhinacanthins from Rhinacanthus nasutus in inhibition against mosquito cytochrome P450 enzymes
由: Rattanawadee Kotewong, et al.
出版: (2018)

Paper-based sol-gel thin films immobilized cytochrome P450 for enzyme activity measurement
由: Nantana Nuchtavorn, et al.
出版: (2020)

An expression of an insect membrane-bound cytochrome P450 CYP6AA3 in the Escherichia coli in relation to insecticide resistance in a malarial vector
由: C. Budriang, et al.
出版: (2018)

Effect of cranberry dietary supplements with different brands on human CYP3A4 enzyme
由: Sompon Wanwimolruk, et al.
出版: (2018)

Regulation of a Cytochrome P450 Gene CYP94B1 by WRKY33 Transcription Factor Controls Apoplastic Barrier Formation in Roots to Confer Salt Tolerance
由: Krishnamurthy, Pannaga, et al.
出版: (2023)