A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines
The reaction of lithio α-chloromethyl phenyl sulfone with imines gave aziridines in good yields. The resulting aziridines were alkylated and underwent the 1,3-dipolar cycloaddition with dimethylacetylene dicarboxylate to give pyrroles in excellent yields. © 1984.
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th-mahidol.305772018-10-12T14:44:38Z A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines Vichai Reutrakul Vichukorn Prapansiri Chitchanun Panyachotipun Mahidol University Biochemistry, Genetics and Molecular Biology Chemistry Pharmacology, Toxicology and Pharmaceutics The reaction of lithio α-chloromethyl phenyl sulfone with imines gave aziridines in good yields. The resulting aziridines were alkylated and underwent the 1,3-dipolar cycloaddition with dimethylacetylene dicarboxylate to give pyrroles in excellent yields. © 1984. 2018-10-12T07:40:15Z 2018-10-12T07:40:15Z 1984-01-01 Article Tetrahedron Letters. Vol.25, No.18 (1984), 1949-1952 10.1016/S0040-4039(01)90084-X 00404039 2-s2.0-0000004487 https://repository.li.mahidol.ac.th/handle/123456789/30577 Mahidol University SCOPUS https://www.scopus.com/inward/record.uri?partnerID=HzOxMe3b&scp=0000004487&origin=inward |
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Biochemistry, Genetics and Molecular Biology Chemistry Pharmacology, Toxicology and Pharmaceutics Vichai Reutrakul Vichukorn Prapansiri Chitchanun Panyachotipun A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines |
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The reaction of lithio α-chloromethyl phenyl sulfone with imines gave aziridines in good yields. The resulting aziridines were alkylated and underwent the 1,3-dipolar cycloaddition with dimethylacetylene dicarboxylate to give pyrroles in excellent yields. © 1984. |
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Mahidol University |
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Mahidol University Vichai Reutrakul Vichukorn Prapansiri Chitchanun Panyachotipun |
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Vichai Reutrakul Vichukorn Prapansiri Chitchanun Panyachotipun |
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Vichai Reutrakul |
title |
A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines |
title_short |
A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines |
title_full |
A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines |
title_fullStr |
A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines |
title_full_unstemmed |
A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines |
title_sort |
new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines |
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2018 |
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https://repository.li.mahidol.ac.th/handle/123456789/30577 |
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