A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines

The reaction of lithio α-chloromethyl phenyl sulfone with imines gave aziridines in good yields. The resulting aziridines were alkylated and underwent the 1,3-dipolar cycloaddition with dimethylacetylene dicarboxylate to give pyrroles in excellent yields. © 1984.

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Main Authors: Vichai Reutrakul, Vichukorn Prapansiri, Chitchanun Panyachotipun
Other Authors: Mahidol University
Format: Article
Published: 2018
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Online Access:https://repository.li.mahidol.ac.th/handle/123456789/30577
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spelling th-mahidol.305772018-10-12T14:44:38Z A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines Vichai Reutrakul Vichukorn Prapansiri Chitchanun Panyachotipun Mahidol University Biochemistry, Genetics and Molecular Biology Chemistry Pharmacology, Toxicology and Pharmaceutics The reaction of lithio α-chloromethyl phenyl sulfone with imines gave aziridines in good yields. The resulting aziridines were alkylated and underwent the 1,3-dipolar cycloaddition with dimethylacetylene dicarboxylate to give pyrroles in excellent yields. © 1984. 2018-10-12T07:40:15Z 2018-10-12T07:40:15Z 1984-01-01 Article Tetrahedron Letters. Vol.25, No.18 (1984), 1949-1952 10.1016/S0040-4039(01)90084-X 00404039 2-s2.0-0000004487 https://repository.li.mahidol.ac.th/handle/123456789/30577 Mahidol University SCOPUS https://www.scopus.com/inward/record.uri?partnerID=HzOxMe3b&scp=0000004487&origin=inward
institution Mahidol University
building Mahidol University Library
continent Asia
country Thailand
Thailand
content_provider Mahidol University Library
collection Mahidol University Institutional Repository
topic Biochemistry, Genetics and Molecular Biology
Chemistry
Pharmacology, Toxicology and Pharmaceutics
spellingShingle Biochemistry, Genetics and Molecular Biology
Chemistry
Pharmacology, Toxicology and Pharmaceutics
Vichai Reutrakul
Vichukorn Prapansiri
Chitchanun Panyachotipun
A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines
description The reaction of lithio α-chloromethyl phenyl sulfone with imines gave aziridines in good yields. The resulting aziridines were alkylated and underwent the 1,3-dipolar cycloaddition with dimethylacetylene dicarboxylate to give pyrroles in excellent yields. © 1984.
author2 Mahidol University
author_facet Mahidol University
Vichai Reutrakul
Vichukorn Prapansiri
Chitchanun Panyachotipun
format Article
author Vichai Reutrakul
Vichukorn Prapansiri
Chitchanun Panyachotipun
author_sort Vichai Reutrakul
title A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines
title_short A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines
title_full A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines
title_fullStr A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines
title_full_unstemmed A new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines
title_sort new method for the synthesis of 2-phenylsulfonylaziridines via the reaction of α-halosulfonyl carbanion to imines
publishDate 2018
url https://repository.li.mahidol.ac.th/handle/123456789/30577
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