Anti-proliferative activity and characterization data on oxadiazole derivatives

by Dukanya, Shanmugam, MK, Rangappa, S, Metri, PK, Mohan, S, Basappa, Rangappa, KS
Published 2022

Synthesis and in vitro antiproliferative activity of diphenyl(sulphonylpiperidin-4-yl)methanol derivatives

by Benaka Prasad, S.B., Vinaya, K., Ananda Kumar, C.S., Swarup, S., Rangappa, K.S.
Published 2014

Synthesis of novel 6-fluoro-3-(4-piperidinyl)-1,2-benzisoxazole derivatives as antiproliferative agents: A structure-activity relationship study

by Benaka Prasad, S.B., Vinaya, K., Ananda Kumar, C.S., Swarup, S., Rangappa, K.S.
Published 2014

Synthesis and in vitro antiproliferative activity of diphenyl(piperidin-4- yl)thioamide methanol derivatives

by Prasad, S.B.B., Vinaya, M.K., Kumar, C.K.S.A., Swarup, S., Rangappa, K.S.
Published 2014

Synthesis and evaluation of 1-benzhydryl-sulfonyl-piperazine derivatives as inhibitors of MDA-MB-231 human breast cancer cell proliferation

by Ananda Kumar, C.S., Nanjunda Swamy, S., Thimmegowda, N.R., Benaka Prasad, S.B., Yip, G.W., Rangappa, K.S.
Published 2015

Synthesis, characterization and evaluation of benzimidazole derivative and its precursors as inhibitors of MDA-MB-231 human breast cancer cell proliferation

by Thimmegowda, N.R., Nanjunda Swamy, S., Ananda Kumar, C.S., Sunil Kumar, Y.C., Chandrappa, S., Yip, G.W., Rangappa, K.S.
Published 2015

Synthesis and in vitro antiproliferative activity of novel 1-benzhydrylpiperazine derivatives against human cancer cell lines

by Kumar, C.S.A., Prasad, S.B.B., Vinaya, K., Chandrappa, S., Thimmegowda, N.R., Kumar, Y.C.S., Swarup, S., Rangappa, K.S.
Published 2014

Synthesis and antiproliferative activity of substituted diazaspiro hydantoins: A structure-activity relationship study

by Ananda Kumar, C.S., Prasad, S.B.B., Vinaya, K., Chandrappa, S., Thimmegowda, N.R., Ranganatha, S.R., Swarup, S., Rangappa, K.S.
Published 2014

Breast cancer stem-like cells are inhibited by diosgenin, a steroidal saponin, by the attenuation of the Wnt β-catenin signaling via the Wnt antagonist secreted frizzled related pr...

by Bhuvanalakshmi, G, Basappa, Laboratory of Chemical Biology, Department of Chemistry, Bangalore University, Bangalore, India, Rangappa, K.S, Dharmarajan, A, Sethi, G, Kumar, A.P, Warrier, S
Published 2020

Anti-cancer activity of novel dibenzo[b,f]azepine tethered isoxazoline derivatives

by Sadashiva, M.P., Basappa, Nanjundaswamy, S., Li, F., Manu, K.A., Sengottuvelan, M., Prasanna, D.S., Anilkumar, N.C., Sethi, G., Sugahara, K., Rangappa, K.S.
Published 2014

The IκB kinase inhibitor ACHP targets the STAT3 signaling pathway in human non-small cell lung carcinoma cells

by Lee, J.H., Mohan, C.D., Basappa, S., Rangappa, S., Chinnathambi, A., Alahmadi, T.A., Alharbi, S.A., Kumar, A.P., Sethi, G., Ahn, K.S., Rangappa, K.S.
Published 2021

Synthesis and characterization of novel 2-amino-chromene-nitriles that target Bcl-2 in acute myeloid leukemia cell lines

by Keerthy H.K., Garg M., Mohan C.D., Madan V., Kanojia D., Shobith R., Nanjundaswamy S., Mason D.J., Bender A., Basappa, Rangappa K.S., Koeffler H.P.
Published 2018

Identification of a novel 1,2 oxazine that can induce apoptosis by targeting NF-κB in hepatocellular carcinoma cells

by Somu, C., Mohan, C.D., Ambekar, S., Dukanya, Rangappa, S., Baburajeev, C.P., Sukhorukov, A., Mishra, S., Shanmugam, M.K., Chinnathambi, A., Awad Alahmadi, T., Alharbi, S.A., Basappa, Rangappa, K.S.
Published 2021

Inhibition of TFF3 enhances sensitivity—and overcomes acquired resistance—to doxorubicin in estrogen receptor-positive mammary carcinoma

by Poh, H.M., Chiou, Y.S., Chong, Q.Y., Chen, R.-M., Rangappa, K.S., Ma, L., Zhu, T., Kumar, A.P., Pandey, V., Basappa, Lee, S.-C., Lobie, P.E.
Published 2021

Brusatol, a nrf2 inhibitor targets stat3 signaling cascade in head and neck squamous cell carcinoma

by Rangappa, K.S., Lee, J.H., Rangappa, S., Mohan, C.D., Basappa, Laboratory of Chemical Biology, Department of Studies in Organic Chemistry, University of Mysore, Manasagangotri, Mysore, 570006, India., Sethi, G., Lin, Z.-X., Ahn, K.S.
Published 2021

Novel 1,3,4-oxadiazole targets STAT3 signaling to induce antitumor effect in lung cancer

by Malojirao, V.H., Girimanchanaika, S.S., Shanmugam, Muthu K., Sherapura, A., Dukanya, Metri, P.K., Vigneshwaran, V., Chinnathambi, A., Alharbi, S.A., Rangappa, S., Mohan, C.D., Basappa, Prabhakar, B.T., Rangappa, K.S.
Published 2021

Trisubstituted-imidazoles induce apoptosis in human breast cancer cells by targeting the oncogenic PI3K/Akt/mTOR signaling pathway

by Mohan C.D., Srinivasa V., Rangappa S., Mervin L., Mohan S., Paricharak S., Baday S., Li F., Shanmugam M.K., Chinnathambi A., Zayed M.E., Alharbi S.A., Bender A., Sethi G., Basappa, Rangappa K.S.
Published 2018

Novel Synthetic Oxazines Target NF-κB in Colon Cancer In Vitro and Inflammatory Bowel Disease In Vivo

by Nirvanappa A.C., Mohan C.D., Rangappa S., Ananda H., Sukhorukov A.Y., Shanmugam M.K., Sundaram M.S., Nayaka S.C., Girish K.S., Chinnathambi A., Zayed M.E., Alharbi S.A., Sethi G., Basappa, Rangappa K.S.
Published 2018

Brusatol suppresses STAT3-driven metastasis by downregulating epithelial-mesenchymal transition in hepatocellular carcinoma

by Lee, J.H., Mohan, C.D., Deivasigamani, A., Jung, Y.Y., Rangappa, S., Basappa, S., Chinnathambi, A., Alahmadi, T.A., Alharbi, S.A., Garg, M., Lin, Z.-X., Rangappa, K.S., Sethi, G., Hui, K.M., Ahn, K.S.
Published 2021

Development of novel triazolo-thiadiazoles from heterogeneous "green" catalysis as protein tyrosine phosphatase 1B inhibitors

by Baburajeev, C.P, Dhananjaya Mohan, C, Ananda, H, Rangappa, S, Fuchs, J.E, Jagadish, S, Sivaraman Siveen, K, Chinnathambi, A, Ali Alharbi, S, Zayed, M.E, Zhang, J, Li, F, Sethi, G, Girish, K.S, Bender, A, Basappa, Rangappa, K.S
Published 2020