Fragment-based approach to the design of 5-chlorouracil-linked-pyrazolo[1, 5-a][1,3,5]triazines as thymidine phosphorylase inhibitors

Fragment-based approach to the design of 5-chlorouracil-linked-pyrazolo[1, 5-a][1,3,5]triazines as thymidine phosphorylase inhibitors

10.1016/j.ejmech.2013.10.022

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Bibliographic Details
Main Authors:	Sun, L., Li, J., Bera, H., Dolzhenko, A.V., Chiu, G.N.C., Chui, W.K.
Other Authors:	PHARMACY
Format:	Article
Published:	2014
Subjects:	5-Chlorouracil-linked-pyrazolo[1,5-a][1,3,5]triazines Fragment-based drug design Mixed-type enzyme inhibition kinetics Thymidine phosphorylase inhibitor
Online Access:	http://scholarbank.nus.edu.sg/handle/10635/105967
Tags:	Add Tag No Tags, Be the first to tag this record!
Institution:	National University of Singapore

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